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Cat. No. Product Name Target Signaling Pathways
TP2073L BigLEN (mouse) acetate

BigLEN (mouse) acetate (501036-69-7 Free base)

GPR Endocrinology/Hormones; GPCR/G Protein
BigLEN (mouse) acetate 是一种有效的、选择性的孤儿 G 蛋白偶联受体 171 (GPR171) 激动剂,Kd 为 ~0.5 nM。
TP2074 BigLEN(rat)

BigLEN (rat)

Potent GPR171 agonist (EC50 = 1.6 nM). ProSAAS-derived peptide. Regulates body weight in mice and promotes the outgrowth of neurites in Neuro2A cells.
TP2073 BigLEN(mouse)

BigLEN (mouse)

GPR171 agonist. ProSAAS-derived neuropeptide. Regulates food intake in mice. Inhibits the release of glutamate onto parvocellular neurons of the paraventricular nucleus in a process dependent upon activation of postsynaptic G proteins.

化合物

BigLEN (mouse) acetate
Cat.No: TP2073L
Synonym: BigLEN (mouse) acetate (501036-69-7 Free base)
Target: GPR
BigLEN(rat)
Cat.No: TP2074
Synonym: BigLEN (rat)
Target:
BigLEN(mouse)
Cat.No: TP2073
Synonym: BigLEN (mouse)
Target:
TargetMol Loading
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